| Alaye ipilẹ | |
| Orukọ ọja | iṣuu soda Cefoperazone + sulfactam iṣuu soda (1: 1/2: 1) |
| Ohun kikọ | Lulú |
| CAS No. | 62893-20-3 693878-84-7 |
| Àwọ̀ | Funfun si ina brown lulú |
| Igbesi aye selifu | ọdun meji 2 |
| Ipele Ipele | Oogun ite |
| Mimo | 99% |
| CAS No. | 62893-20-3 |
| Package | 10kg / ilu |
Apejuwe
Apejuwe:
Cefoperzone sodium + sulbactam sodium (1: 1/2: 1) jẹ iṣẹ-ṣiṣe obi, inhibitor β-lactamase laipe ti a ṣe bi 1: 1 ọja apapo pẹlu cefoperazone. Gẹgẹbi clavulanic acid, aṣoju akọkọ ti iru yii lati ṣe afihan, sulbactam ṣe imudara imunadoko ti awọn egboogi β-lactam lodi si awọn igara sooro.
Lilo:
Oludena β-lactamase ologbele-sintetiki. O ti wa ni lilo ni apapo pẹlu β-lactam egboogi bi antibacterial.
Iyọ iṣuu soda Cefoperazone jẹ oogun apakokoro cephalosporin fun idinamọ ti gbigba rMrp2-mediated [3H] E217βG pẹlu IC50 ti 199 μM. Àfojúsùn: Cefoperazone Antibacterial jẹ aibikita, semisynthetic, spekitiriumu gbooro, aporo aporo cephalosporin parenteral fun iṣakoso iṣan tabi iṣan inu. Lẹhin iṣakoso iṣọn-ẹjẹ ti 2 g ti Cefoperazone, awọn ipele ninu omi ara wa lati 202μg/mL si 375 μg/mL da lori akoko iṣakoso oogun. Lẹhin abẹrẹ inu iṣan ti 2 g ti Cefoperazone, apapọ ipele omi ara ti o ga julọ jẹ 111 μg/mL ni awọn wakati 1.5. Ni awọn wakati 12 lẹhin iwọn lilo, awọn ipele omi ara tumọ si tun jẹ 2 si 4 μg/mL. Cefoperazone jẹ 90% ti sopọ mọ awọn ọlọjẹ ara.








